SCHEMBL6946442

SCHEMBL6946442

O=C(O)CC(=O)c1cccc2[nH]c(Cc3ccccc3)nc12

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.49
GRIN1 Q05586 1/20 0.49
GAA P10253 2/20 0.49
HTR6 P50406 2/20 0.48
BRD4 O60885 1/20 0.45
CREBBP Q92793 1/20 0.45
PKM P14618 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TSHR P16473 1/20 0.43
PARP1 P09874 4/20 0.42
DHODH Q02127 2/20 0.42
RNASEH1 O60930 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946473 0.88 NPC1 (0.50) GAABRD4CREBBPPARP1DHODH
SCHEMBL6951804 0.84 HTR6 (0.52) GRIN2BGRIN1GAAHTR6BRD4
SCHEMBL6950138 0.79 KMT2A (0.49) GRIN2BGRIN1GAAPKMSMN1; SMN2
SCHEMBL6948942 0.77 BRD4 (0.50) GAABRD4CREBBPSMN1; SMN2PARP1
SCHEMBL6949839 0.77 CHEK1 (0.50) BRD4CREBBPPARP1
SCHEMBL6948419 0.76 PARP1 (0.45) GAABRD4CREBBPPARP1RNASEH1
SCHEMBL9540471 0.76 GRIN2B (0.77) GRIN2BGRIN1GAAHTR6PKM
SCHEMBL6542830 0.74 GAA (0.60) GRIN2BGRIN1GAAHTR6PKM
SCHEMBL6948954 0.74 NPC1 (0.55) PARP1DHODHRNASEH1
SCHEMBL6946441 0.73 PARP1 (0.48) GAABRD4CREBBPPARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936218-B1 BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARM CO LTD (JP) 2003-04-02 EP disclosed
US-6387938-B1 Benzimidazole derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-05-14 US disclosed
EP-0936218-A1 NOVEL BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1999-08-18 EP disclosed