SCHEMBL6947355

SCHEMBL6947355

CC(C)C[C@@H](C(=O)NN)[C@@H](C(=O)NOC1CCCCO1)C(/C=C/c1ccccc1)(CCc1c[nH]c2ccccc12)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 4/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SIRT2 Q8IXJ6 2/20 0.35
MC3R P41968 1/20 0.35
HPGD P15428 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC3 O15379 4/20 0.34
HDAC4 P56524 4/20 0.34
HDAC1 Q13547 4/20 0.34
HDAC7 Q8WUI4 4/20 0.34
HDAC2 Q92769 4/20 0.34
HDAC10 Q969S8 4/20 0.34
HDAC11 Q96DB2 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945554 0.87 ADAM17 (0.33) ALDH1A1MMP2MMP9
SCHEMBL6946721 0.87 ADAM17 (0.32) MMP2MMP9
SCHEMBL8097980 0.86 GPR88 (0.31)
SCHEMBL6942184 0.86 ECE1 (0.46) ECE1ALDH1A1SIRT2HPGDMMP2
SCHEMBL7937084 0.85 ALDH1A1 (0.33) ALDH1A1MMP2MMP9
SCHEMBL6945788 0.85 ADAM17 (0.31) MMP2MMP9
SCHEMBL6942507 0.85 FKBP1A (0.32) MMP2MMP9
SCHEMBL6943876 0.85 ADAM17 (0.31) MMP2MMP9
SCHEMBL6942209 0.85 ADAM17 (0.33) ALDH1A1MMP2MMP9
SCHEMBL8111706 0.85 ADAM17 (0.33) ALDH1A1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed