SCHEMBL6947640

SCHEMBL6947640

O=CC(C(=O)C(=O)O)c1ccc2cc(Cc3ccc(F)cc3)[nH]c2c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.39
DDO Q99489 1/20 0.36
PIN1 Q13526 4/20 0.36
EIF4A3 P38919 1/20 0.34
PDE2A O00408 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALB P02768 1/20 0.32
IL2 P60568 1/20 0.32
BRS3 P32247 1/20 0.32
ITK Q08881 1/20 0.32
F2 P00734 1/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950558 0.74 ITK (0.39) DAODDOPIN1ITKF2
SCHEMBL6990951 0.74 DAO (0.49) DAODDOPIN1F2
Hydroxyamine SCHEMBL4796191 0.73 NR4A2 (0.46) DAODDOPIN1ITKF2
SCHEMBL5132984 0.70 HDAC6 (0.51) PIN1ITK
SCHEMBL6994150 0.69 DAO (0.44) DAODDOITK
SCHEMBL6943878 0.69 DAO (0.40) DAODDOTDP1F2
SCHEMBL6992345 0.69 SIGMAR1 (0.46) DAODDO
SCHEMBL6949840 0.69 F2 (0.47) DAOPIN1TDP1F2PPARG
SCHEMBL6947529 0.68 NR4A2 (0.56)
SCHEMBL6994522 0.67 LOXL2 (0.53) F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed