SCHEMBL6949795

SCHEMBL6949795

CCOC(=O)c1c(-c2ccc(F)cc2)nc(C)c(C(=O)OC)c1C(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.50
ALDH1A1 P00352 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GCGR P47871 1/20 0.49
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
SLC26A6 Q9BXS9 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
LMNA P02545 1/20 0.44
PTGS2 P35354 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
CASP3 P42574 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8178136 0.84 GCGR (0.64) ALDH1A1L3MBTL1GCGRPOLBGAA
SCHEMBL6960560 0.84 GCGR (0.49) ADORA3ALDH1A1L3MBTL1GCGRNPC1
SCHEMBL6949885 0.83 ADORA3 (0.46) ADORA3ALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL6956758 0.82 ADORA3 (0.46) ADORA3ALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL9737768 0.82 GCGR (0.64) ALDH1A1L3MBTL1GCGRPOLBGAA
SCHEMBL15481445 0.79 ALDH1A1 (0.47) ADORA3ALDH1A1L3MBTL1GCGRGAA
SCHEMBL3206 0.78 GCGR (0.47) ADORA3ALDH1A1L3MBTL1GCGRPOLB
SCHEMBL7566003 0.78 ALDH1A1 (0.57) ADORA3ALDH1A1L3MBTL1POLBGAA
SCHEMBL13482768 0.77 GCGR (0.64) ALDH1A1L3MBTL1GCGRPOLBGAA
SCHEMBL2211 0.77 ALDH1A1 (0.47) ADORA3ALDH1A1L3MBTL1GCGRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325130-B1 Substituted pyridines BAYER AG (DE) 2003-11-05 EP disclosed
EP-1123925-A1 Process for preparation of substituted pyridines BAYER AG (DE) 2001-08-16 EP disclosed
EP-1123924-A1 Substituted pyridines as HMG-COA reductase inhibitors BAYER AG (DE) 2001-08-16 EP disclosed
CN-1274719-A Process for preparation of substituted pyridine compound BAYER AG (DE) 2000-11-29 CN disclosed
CN-1055684-C Process for preparing substituted pyridine compounds BAYER AG (DE) 2000-08-23 CN disclosed
US-5401746-A FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND HMG-COA REDUCTASE BAYER AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
US-5006530-A Certain 7-[2,6-diisopropyl-4-phenyl-5-lower alkoxymethyl-pyrid-3-yl]-3,5-dihydroxy-6-enoates and derivatives useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1991-04-09 US disclosed
CN-1034364-A Substituted pyridines and process for their preparation BAYER AG (DE) 1989-08-02 CN disclosed
EP-0325130-A2 Substituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed