SCHEMBL6950602

SCHEMBL6950602

O=C(O)C(=O)CC(=O)c1cc(Cc2ccccc2)cc(-c2cnccn2)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 6/20 0.47
FEN1 P39748 6/20 0.47
PTPN1 P18031 4/20 0.45
PIM2 Q9P1W9 2/20 0.43
HAO1 Q9UJM8 4/20 0.41
PLOD2 O00469 1/20 0.40
PIM1 P11309 1/20 0.40
WNT3A P56704 1/20 0.39
MAOA P21397 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949374 0.84 PTPN1 (0.45) ERCC5FEN1PTPN1HAO1PLOD2
SCHEMBL7077395 0.82 WNT3A (0.43) PIM2PLOD2PIM1WNT3ASMN1; SMN2
SCHEMBL7073904 0.81 TBXAS1 (0.52) ERCC5FEN1PTPN1PLOD2
SCHEMBL7667672 0.80 PIM2 (0.41) ERCC5FEN1PTPN1PIM2HAO1
SCHEMBL6947604 0.78 ERCC5 (0.61) ERCC5FEN1PTPN1HAO1
SCHEMBL7667601 0.75 PIM2 (0.56) PIM2PIM1
SCHEMBL6949384 0.75 ERCC5 (0.46) ERCC5FEN1PTPN1HAO1SMN1; SMN2
SCHEMBL6945686 0.75 ERCC5 (0.46) ERCC5FEN1PTPN1HAO1
SCHEMBL6948009 0.74 PTPN1 (0.57) ERCC5FEN1PTPN1HAO1PLOD2
SCHEMBL6940911 0.74 PTPN1 (0.72) ERCC5FEN1PTPN1HAO1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed