SCHEMBL7667672

SCHEMBL7667672

CN(C)c1cncc(-c2cc(Cc3ccccc3)cc(C(=O)CC(=O)C(=O)O)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIM2 Q9P1W9 2/20 0.41
ERCC5 P28715 4/20 0.40
FEN1 P39748 4/20 0.40
PTPN1 P18031 4/20 0.39
BRAF P15056 5/20 0.38
HAO1 Q9UJM8 3/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
BRD4 O60885 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950602 0.80 ERCC5 (0.47) PIM2ERCC5FEN1PTPN1HAO1
SCHEMBL7667601 0.79 PIM2 (0.56) PIM2PIM1
SCHEMBL6946034 0.75 PTPN1 (0.53) ERCC5FEN1PTPN1HAO1
SCHEMBL6945686 0.75 ERCC5 (0.46) ERCC5FEN1PTPN1HAO1
SCHEMBL6947604 0.74 ERCC5 (0.61) ERCC5FEN1PTPN1HAO1
SCHEMBL7073904 0.72 TBXAS1 (0.52) ERCC5FEN1PTPN1
SCHEMBL6949748 0.71 ERCC5 (0.53) ERCC5FEN1PTPN1HAO1
SCHEMBL7082801 0.70 LMNA (0.44) BRAFCYP11B1CYP11B2
SCHEMBL6949374 0.68 PTPN1 (0.45) ERCC5FEN1PTPN1HAO1
SCHEMBL6948238 0.68 PTPN1 (0.44) ERCC5FEN1PTPN1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed