SCHEMBL695644

SCHEMBL695644

Cc1nn(CC(F)(F)F)c(N2CCCC2C(=O)O)c1S(C)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
LMNA P02545 2/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KEAP1 Q14145 2/20 0.33
POLB P06746 1/20 0.32
AADAT Q8N5Z0 1/20 0.32
SYK P43405 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697456 0.89 PEPD (0.36) KMT2AALDH1A1LMNAPOLBAADAT
SCHEMBL696511 0.88 KMT2A (0.33) KMT2AMAPTLMNACYP2C19HSD17B10
SCHEMBL695772 0.79 ALDH1A1 (0.41) ALDH1A1HPGDLMNAKEAP1
SCHEMBL695240 0.77 CNR2 (0.41) KMT2AALDH1A1LMNACYP2C19SYK
SCHEMBL696236 0.77 ADORA2A (0.35) LMNASMN1; SMN2
SCHEMBL695637 0.70 FKBP1A (0.42) MAPTALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL696054 0.68 ACE (0.37) ALDH1A1HPGDLMNAKEAP1
SCHEMBL694119 0.68 CNR2 (0.38) KMT2AALDH1A1LMNACYP2C19POLB
SCHEMBL696423 0.67 MCHR1 (0.42) KMT2AMAPTALDH1A1CYP2C19
SCHEMBL696225 0.66 KMT2A (0.37) KMT2AMAPTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed