SCHEMBL695772

SCHEMBL695772

Cc1nn(CCc2ccccc2)c(N2CCCC2C(=O)O)c1S(C)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
ACE P12821 5/20 0.39
MMP1 P03956 1/20 0.39
MMP7 P09237 1/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP13 P45452 1/20 0.39
FKBP1A P62942 4/20 0.38
KEAP1 Q14145 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695637 0.91 FKBP1A (0.42) ALDH1A1HPGDMMP1MMP7MMP8
SCHEMBL696054 0.89 ACE (0.37) ALDH1A1HPGDACEMMP1MMP7
SCHEMBL695528 0.86 CCR4 (0.36) ALDH1A1HPGDACEMMP1MMP7
SCHEMBL3719340 0.82 RAB9A (0.37) KEAP1RAB9ALMNA
SCHEMBL3724272 0.81 FKBP1A (0.37) ALDH1A1FKBP1A
SCHEMBL696519 0.80 FKBP1A (0.40) ALDH1A1HPGDMMP1MMP7MMP8
SCHEMBL695644 0.79 KMT2A (0.35) ALDH1A1HPGDKEAP1LMNA
SCHEMBL696150 0.78 FKBP1A (0.40) ALDH1A1HPGDMMP1MMP7MMP8
SCHEMBL696225 0.73 KMT2A (0.37) ALDH1A1LMNA
SCHEMBL695240 0.72 CNR2 (0.41) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed