SCHEMBL697456

SCHEMBL697456

COC(=O)C1CCCN1c1c(S(C)(=O)=O)c(C)nn1CC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PEPD P12955 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
MCHR1 Q99705 1/20 0.34
FKBP1A P62942 2/20 0.33
SCN9A Q15858 2/20 0.32
MMP2 P08253 1/20 0.32
ANPEP P15144 1/20 0.32
FPR2 P25090 1/20 0.32
LMNA P02545 2/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
ULK1 O75385 1/20 0.31
AADAT Q8N5Z0 1/20 0.31
POLB P06746 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695644 0.89 KMT2A (0.35) LMNASMN1; SMN2ALDH1A1KMT2AAADAT
SCHEMBL696236 0.88 ADORA2A (0.35) PEPDADORA2AADORA1MCHR1SCN9A
SCHEMBL695637 0.80 FKBP1A (0.42) FKBP1ASCN9ARAB9ASMN1; SMN2ALDH1A1
SCHEMBL696423 0.79 MCHR1 (0.42) ADORA2AADORA1MCHR1FPR2ALDH1A1
SCHEMBL696511 0.77 KMT2A (0.33) LMNAKMT2AAADATPOLB
SCHEMBL696519 0.69 FKBP1A (0.40) FKBP1ASCN9ARAB9ASMN1; SMN2ALDH1A1
SCHEMBL694464 0.69 MCHR1 (0.41) ADORA2AADORA1MCHR1FPR2LMNA
SCHEMBL695772 0.69 ALDH1A1 (0.41) FKBP1ALMNARAB9AALDH1A1
SCHEMBL696114 0.68 DRD2 (0.38) FKBP1AFPR2LMNAALDH1A1KMT2A
SCHEMBL696150 0.68 FKBP1A (0.40) FKBP1ARAB9ASMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed