SCHEMBL696150

SCHEMBL696150

COC(=O)C1CCCN1c1c(S(=O)(=O)c2ccccc2Cl)c(C)nn1CCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 3/20 0.40
LTA4H P09960 2/20 0.38
ALDH1A1 P00352 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CTSS P25774 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
MMP1 P03956 1/20 0.35
MMP7 P09237 1/20 0.35
MMP8 P22894 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695528 0.92 CCR4 (0.36) FKBP1AALDH1A1NPC1RAB9AHPGD
SCHEMBL696114 0.88 DRD2 (0.38) FKBP1AALDH1A1CTSSMAPT
SCHEMBL695637 0.87 FKBP1A (0.42) FKBP1ALTA4HALDH1A1NPC1RAB9A
SCHEMBL3724272 0.87 FKBP1A (0.37) FKBP1AALDH1A1
SCHEMBL696519 0.84 FKBP1A (0.40) FKBP1ALTA4HALDH1A1NPC1RAB9A
SCHEMBL3719340 0.82 RAB9A (0.37) RAB9ACCR4
SCHEMBL696304 0.82 FKBP1A (0.39) FKBP1ALTA4HCTSSNPSR1MAPT
SCHEMBL695533 0.81 OPRM1 (0.41) FKBP1AALDH1A1CTSSNPSR1MAPT
SCHEMBL696225 0.80 KMT2A (0.37) ALDH1A1MAPTSMN1; SMN2
SCHEMBL695720 0.79 CTSS (0.37) FKBP1ACTSSNPSR1USP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed