SCHEMBL6958387

SCHEMBL6958387

O=C(Nc1cnccn1)N(S)CCc1c(F)cccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 3/20 0.46
GSK3B P49841 3/20 0.46
CDK5 Q00535 3/20 0.46
PRKD3 O94806 2/20 0.46
MAP4K4 O95819 2/20 0.46
CLK2 P49760 2/20 0.46
PRKAA1 Q13131 2/20 0.46
DYRK1A Q13627 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
CDC7 O00311 1/20 0.46
AURKA O14965 1/20 0.46
CDK1 P06493 1/20 0.46
CSF1R P07333 1/20 0.46
CDK2 P24941 1/20 0.46
MAPK1 P28482 1/20 0.46
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
CSNK1D P48730 1/20 0.46
MAPK12 P53778 1/20 0.46
CSNK2A1 P68400 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958381 0.72 ALDH1A1 (0.47) GSK3AGSK3BCDK5PRKD3MAP4K4
SCHEMBL8685471 0.68 KMT2A (0.43) GSK3AGSK3BCDK5PRKD3MAP4K4
SCHEMBL11537230 0.64 KMT2A (0.42) KMT2AKDM4EMEN1THRBNPC1
SCHEMBL25097159 0.63 KMT2A (0.54) KMT2ATSHRGAAKDM4EMEN1
SCHEMBL3795739 0.63 CDK5 (1.00) GSK3AGSK3BCDK5PRKD3MAP4K4
SCHEMBL6625255 0.63 GAA (0.50) KMT2ATSHRGAAKDM4EMEN1
SCHEMBL5381046 0.62 KDM4E (0.69) GSK3AGSK3BCDK5PRKD3MAP4K4
SCHEMBL9579797 0.62 CNR1 (0.40) GSK3AGSK3BCDK5PRKD3MAP4K4
SCHEMBL8495201 0.62 RAB9A (0.51) KMT2AGAAKDM4EMEN1POLB
SCHEMBL24967599 0.61 SMN1; SMN2 (0.61) GSK3AGSK3BCDK5PRKD3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5714503-A Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 1998-02-03 US disclosed
US-5658907-A THIOUREA VIRICIDES MEDIVIR A/B (SE) 1997-08-19 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
WO-1993003022-A1 COMPOUNDS AND METHODS FOR INHIBITION OF HIV AND RELATED VIRUSES MEDIVIR AB (SE) 1993-02-18 WO disclosed