SCHEMBL6959376

SCHEMBL6959376

CC(C)(C)OC(=O)CN1C(=O)CN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.41
BCL2 P10415 1/20 0.40
BECN1 Q14457 1/20 0.40
BCHE P06276 1/20 0.40
P2RX4 Q99571 1/20 0.40
HPGD P15428 1/20 0.39
HTR1A P08908 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
XIAP P98170 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
ATM Q13315 1/20 0.38
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959586 0.85 HDAC1 (0.49) HDAC1HDAC6P2RX4XIAP
SCHEMBL7140109 0.79 L3MBTL1 (0.45) L3MBTL1BCHEP2RX4HPGDHTR1A
SCHEMBL6972375 0.78 KDM4E (0.43) L3MBTL1BCHEP2RX4HPGDHTR1A
SCHEMBL6955643 0.77 L3MBTL1 (0.46) L3MBTL1HPGDALDH1A1NPC1RAB9A
SCHEMBL6969043 0.77 DRD3 (0.47) L3MBTL1BCHEP2RX4HPGDHTR1A
SCHEMBL6964416 0.74 DRD2 (0.50) L3MBTL1HPGDHTR1ATDP1ALDH1A1
SCHEMBL6959609 0.74 AVPR2 (0.50)
SCHEMBL6972297 0.72 ALDH1A1 (0.46) L3MBTL1TDP1ALDH1A1MAPTLMNA
SCHEMBL8421386 0.71 CES1 (0.53) BCHEHPGDTDP1ALDH1A1ATM
SCHEMBL6960672 0.71 L3MBTL1 (0.46) L3MBTL1TDP1ALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed