SCHEMBL6960286

SCHEMBL6960286

Cc1nn(-c2ccccc2)cc1N(Cc1cccc(C#N)c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.38
PTGES O14684 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
MEP1A Q16819 1/20 0.36
MEP1B Q16820 1/20 0.36
SLC16A3 O15427 1/20 0.36
SLC16A1 P53985 1/20 0.36
MCTS1 Q9ULC4 1/20 0.36
MCL1 Q07820 1/20 0.36
ALKBH1 Q13686 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
PDK1 Q15118 1/20 0.35
CACNA2D1 P54289 1/20 0.35
ABCB1 P08183 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971033 0.87 NR3C1 (0.42) NR3C1MEP1AMEP1BALKBH1PDK1
SCHEMBL6972367 0.83 ALKBH1 (0.42) PTGESCHRM2CHRM1CHRM3MEP1A
SCHEMBL6963537 0.82 PTGES (0.38) NR3C1PTGESCHRM2CHRM1CHRM3
SCHEMBL6955000 0.80 PTGES (0.38) NR3C1PTGESCHRM2CHRM1CHRM3
SCHEMBL15362537 0.79 HTT (0.41) MCL1HTR2CSLC6A4CACNA2D1
SCHEMBL6955361 0.79 PTGES (0.37) PTGESCHRM2CHRM1CHRM3MEP1A
SCHEMBL1010216 0.73 MEP1A (0.50) PTGESCHRM2CHRM1CHRM3MEP1A
SCHEMBL320434 0.72 MEP1A (0.49) PTGESCHRM2CHRM1CHRM3MEP1A
SCHEMBL6964182 0.70 MEP1A (0.38) PTGESCHRM2CHRM1CHRM3MEP1A
SCHEMBL1010217 0.70 MEP1A (0.47) PTGESCHRM2CHRM1CHRM3MEP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed