SCHEMBL6972367

SCHEMBL6972367

CC(C)(C)OC(=O)N(Cc1cccc(C#N)c1)c1cnn(-c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALKBH1 Q13686 1/20 0.42
CHRM2 P08172 2/20 0.41
CHRM1 P11229 2/20 0.41
CHRM3 P20309 2/20 0.41
PTGES O14684 1/20 0.38
MEP1A Q16819 1/20 0.37
MEP1B Q16820 1/20 0.37
GRM5 P41594 1/20 0.37
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
MCL1 Q07820 1/20 0.36
PDK1 Q15118 1/20 0.36
VNN1 O95497 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
ABCB1 P08183 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966037 0.86 ALKBH1 (0.43) ALKBH1CHRM2CHRM1CHRM3MEP1A
SCHEMBL6960286 0.83 NR3C1 (0.38) ALKBH1CHRM2CHRM1CHRM3PTGES
SCHEMBL6955000 0.81 PTGES (0.38) ALKBH1CHRM2CHRM1CHRM3PTGES
SCHEMBL6963537 0.81 PTGES (0.38) ALKBH1CHRM2CHRM1CHRM3PTGES
SCHEMBL31456982 0.81 ITGB1 (0.41) CHRM2CHRM1CHRM3MCL1MEN1
SCHEMBL6955361 0.80 PTGES (0.37) ALKBH1CHRM2CHRM1CHRM3PTGES
SCHEMBL1010216 0.76 MEP1A (0.50) CHRM2CHRM1CHRM3PTGESMEP1A
SCHEMBL24467961 0.73 GPR119 (0.37) ALKBH1FNTAFNTB
SCHEMBL29741623 0.73 KCNJ1 (0.38) ALKBH1FNTAFNTB
SCHEMBL320434 0.73 MEP1A (0.49) CHRM2CHRM1CHRM3PTGESMEP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed