SCHEMBL6960341

SCHEMBL6960341

CC(C)c1nc(C=O)n(Cc2ccccn2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 8/20 0.35
GRIN1 Q05586 5/20 0.35
GRIN2B Q13224 5/20 0.35
BRD4 O60885 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GFER P55789 1/20 0.32
RIPK3 Q9Y572 1/20 0.32
ALOX5AP P20292 1/20 0.32
P2RX7 Q99572 1/20 0.32
P2RX3 P56373 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967288 0.92 GRIN1 (0.40) S1PR3GRIN1GRIN2BBRD4KDM4E
SCHEMBL6973368 0.89 ALDH1A1 (0.34) BRD4KDM4EALDH1A1LMNAALOX5AP
SCHEMBL6973236 0.88 ALDH1A1 (0.35) S1PR3GRIN1GRIN2BBRD4ALDH1A1
SCHEMBL7084152 0.87 S1PR3 (0.34) S1PR3GRIN1GRIN2BKDM4EALDH1A1
SCHEMBL7084149 0.87 S1PR3 (0.34) S1PR3GRIN1GRIN2BKDM4EALDH1A1
SCHEMBL6973903 0.84 GRIN1 (0.38) GRIN1GRIN2BBRD4KDM4EALDH1A1
SCHEMBL7078209 0.83 S1PR3 (0.34) S1PR3GRIN1GRIN2BBRD4KDM4E
SCHEMBL6973511 0.83 S1PR3 (0.36) S1PR3GRIN1GRIN2BKDM4EALDH1A1
SCHEMBL6972005 0.82 VDR (0.32) GRIN1GRIN2B
SCHEMBL6973761 0.81 CFTR (0.44) S1PR3KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed