SCHEMBL6973236

SCHEMBL6973236

CC(C)c1nc(C=O)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
AGTR1 P30556 1/20 0.35
NOX4 Q9NPH5 4/20 0.34
P2RX3 P56373 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
VDR P11473 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRA5 P31644 1/20 0.33
BRD4 O60885 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
S1PR3 Q99500 1/20 0.32
TP53 P04637 1/20 0.32
CYBB P04839 1/20 0.32
CYP3A4 P08684 1/20 0.32
NOX1 Q9Y5S8 1/20 0.32
ALOX5AP P20292 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973903 0.92 GRIN1 (0.38) ALDH1A1AGTR1NOX4P2RX3GRIN1
SCHEMBL6973368 0.89 ALDH1A1 (0.34) ALDH1A1NOX4MEN1KMT2AGABRA1
SCHEMBL6960341 0.88 S1PR3 (0.35) ALDH1A1P2RX3GRIN1GRIN2BBRD4
SCHEMBL6969160 0.87 ADRA1D (0.32) ALDH1A1AGTR1NOX4P2RX3MEN1
SCHEMBL6969157 0.87 ADRA1D (0.32) ALDH1A1AGTR1NOX4P2RX3MEN1
SCHEMBL6967288 0.84 GRIN1 (0.40) NOX4GRIN1GRIN2BKMT2ABRD4
SCHEMBL6967722 0.83 TDP1 (0.34) MEN1KMT2AVDRTDP1
SCHEMBL6975001 0.83 ALDH1A1 (0.33) ALDH1A1AGTR1NOX4P2RX3GRIN1
SCHEMBL6976953 0.83 ALDH1A1 (0.33) ALDH1A1AGTR1NOX4P2RX3GRIN1
SCHEMBL6973761 0.81 CFTR (0.44) ALDH1A1MEN1KMT2AS1PR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed