SCHEMBL6962482

SCHEMBL6962482

Nc1cccc(CCN(C(=O)C(F)(F)F)c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
GRM2 Q14416 1/20 0.41
GRM3 Q14832 1/20 0.41
CYP19A1 P11511 1/20 0.40
MLYCD O95822 3/20 0.38
SIGMAR1 Q99720 2/20 0.37
CES1 P23141 1/20 0.36
OPRK1 P41145 1/20 0.36
PBRM1 Q86U86 1/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961364 0.84 MAOA (0.54) MAOAMAOBMEN1KMT2AGRM2
SCHEMBL6955778 0.80 ALDH1A1 (0.48) SMN1; SMN2MEN1CYP2C9CYP2C19KMT2A
SCHEMBL6956921 0.75 GRIN2D (0.45) MAOAMAOBMEN1CYP2C19KMT2A
SCHEMBL31211648 0.72 SMN1; SMN2 (0.59) SMN1; SMN2MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL3441981 0.71 HSD11B1 (0.53) MEN1KMT2A
SCHEMBL16366240 0.70 GYS1 (0.39) MAOAMAOBGRM2GRM3CYP19A1
SCHEMBL1205533 0.70 MAOA (0.49) MAOAMAOBMEN1KMT2AGRM2
SCHEMBL11696798 0.69 MLYCD (0.49) MEN1KMT2AMLYCDCES1NPC1
SCHEMBL27770722 0.69 MAOA (0.51) MAOAMAOBMEN1KMT2AGRM2
SCHEMBL31211569 0.69 NPC1 (0.60) SMN1; SMN2MEN1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed