SCHEMBL6955778

SCHEMBL6955778

O=C(N(CCc1cccc([N+](=O)[O-])c1)c1ccccc1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
LMNA P02545 2/20 0.48
HTT P42858 2/20 0.47
PKM P14618 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
MAPT P10636 1/20 0.45
ATM Q13315 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HPGD P15428 2/20 0.44
SIGMAR1 Q99720 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967315 0.85 KCNH2 (0.58) ALDH1A1LMNAHTTSMN1; SMN2RAB9A
SCHEMBL6962482 0.80 MAOA (0.47) ALDH1A1HTTSMN1; SMN2RAB9ANPC1
SCHEMBL6963390 0.78 ALDH1A1 (0.59) ALDH1A1LMNAHTTPKMKDM4E
SCHEMBL3441758 0.74 PYCR1 (0.53) ALDH1A1LMNAHTTSMN1; SMN2RAB9A
SCHEMBL16366561 0.73 ALDH1A1 (0.50) ALDH1A1LMNAHTTPKMSMN1; SMN2
SCHEMBL15921150 0.73 TSHR (0.65) ALDH1A1LMNAHTTSMN1; SMN2RAB9A
SCHEMBL1204373 0.73 ALDH1A1 (0.52) ALDH1A1LMNASMN1; SMN2CYP1A2CYP2D6
SCHEMBL1204376 0.73 ALDH1A1 (0.52) ALDH1A1LMNASMN1; SMN2CYP1A2CYP2D6
SCHEMBL14267707 0.71 SIGMAR1 (0.48) ALDH1A1LMNAHTTSMN1; SMN2RAB9A
SCHEMBL1435064 0.71 CRHBP (0.55) ALDH1A1LMNAPKMSMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed