SCHEMBL6962674

SCHEMBL6962674

CC(C)c1nc(C=O)n(Cc2cccnc2)c1Sc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
RAD1 O60671 1/20 0.36
MAPT P10636 1/20 0.36
CFTR P13569 1/20 0.36
APEX1 P27695 1/20 0.36
CASP6 P55212 1/20 0.36
KMT2A Q03164 1/20 0.36
RAD51 Q06609 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
GOPC Q9HD26 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 1/20 0.36
GABRA1 P14867 2/20 0.35
GABRA5 P31644 2/20 0.35
PDE5A O76074 1/20 0.35
TBXAS1 P24557 2/20 0.35
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970262 0.88 GRIN1 (0.41)
SCHEMBL6970594 0.88 ALDH1A1 (0.40) ALDH1A1KDM4EKMT2ATDP1GABRA1
SCHEMBL6964826 0.88 VDR (0.36) ALOX5APALDH1A1KDM4EMAPTKMT2A
SCHEMBL6967171 0.88 GRIN1 (0.41) ALDH1A1PKM
SCHEMBL6968924 0.88 GABRA5 (0.37) ALOX5APALDH1A1KMT2ATDP1GABRA1
SCHEMBL8099988 0.87 ALOX5AP (0.35) ALOX5APALDH1A1KDM4ERAD1MAPT
SCHEMBL8099986 0.87 ALOX5AP (0.35) ALOX5APALDH1A1KDM4ERAD1MAPT
SCHEMBL6973483 0.85 MAPT (0.37) ALDH1A1KDM4EMAPTKMT2ATDP1
SCHEMBL6972848 0.82 TLR7 (0.38) ALOX5APALDH1A1KDM4EMAPK1GABRA1
SCHEMBL7081083 0.82 ALOX5AP (0.37) ALOX5APALDH1A1KDM4EMAPK1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed