SCHEMBL6962804

SCHEMBL6962804

Cc1nc2ccc(Sc3cccc4cnccc34)cc2n1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.47
DHFR P00374 1/20 0.42
CYP11B2 P19099 1/20 0.41
GALR3 O60755 2/20 0.40
NR2F2 P24468 2/20 0.40
RAB9A P51151 1/20 0.40
DCTPP1 Q9H773 2/20 0.39
BRD4 O60885 3/20 0.39
SPHK1 Q9NYA1 1/20 0.38
THRB P10828 1/20 0.37
TP53 P04637 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974563 0.76 KDM4E (0.41) CYP11B2RAB9ADCTPP1
SCHEMBL6968731 0.72 KDM4E (0.41) CYP11B2RAB9AROCK2ROCK1
SCHEMBL8358073 0.70 KDR (0.44)
SCHEMBL615476 0.70 TNF (0.68) TNFDHFRGALR3NR2F2RAB9A
SCHEMBL317642 0.70 DCTPP1 (0.70) TNFDHFRGALR3NR2F2RAB9A
SCHEMBL14340743 0.70 LMNA (0.48) DHFRRAB9A
SCHEMBL6957957 0.70 ALDH1A1 (0.36) RAB9ATP53
Hydrochloric Acid SCHEMBL7085899 0.69 TYMS (0.46) RAB9A
SCHEMBL6966199 0.68 HDAC6 (0.42) GALR3NR2F2ROCK2ROCK1
SCHEMBL6969044 0.68 KDM4E (0.36) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed