SCHEMBL6964916

SCHEMBL6964916

CC(=O)OCCOC(C)c1nc(C(C)C)c(Sc2ccccc2)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33
TUBB3 Q13509 2/20 0.33
TUBB2A Q13885 2/20 0.33
TUBB8 Q3ZCM7 2/20 0.33
TUBA3E Q6PEY2 2/20 0.33
TUBA1A Q71U36 2/20 0.33
TUBA1C Q9BQE3 2/20 0.33
TUBB6 Q9BUF5 2/20 0.33
TUBB2B Q9BVA1 2/20 0.33
TUBB1 Q9H4B7 2/20 0.33
DHFR P00374 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086334 0.89 DHFR (0.32) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL7082473 0.88 SLC6A9 (0.34) CA2CA4L3MBTL1ALDH1A1
SCHEMBL6968877 0.88 SLC6A9 (0.36) DHFRKMT2AMEN1CYP1A2CYP2C9
SCHEMBL7080480 0.85 DHFR (0.36) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL6962840 0.85
SCHEMBL7085474 0.85 CYP2C9 (0.38) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL6966250 0.84 TUBB4A (0.37) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL6975782 0.83 CDK5 (0.33) CYP1A2CYP2C9CYP2C19ALDH1A1CDK5
SCHEMBL7080029 0.83 PTPRA (0.34) CYP1A2ALDH1A1
SCHEMBL6973132 0.81 LMNA (0.34) KMT2AMEN1CYP1A2L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed