SCHEMBL6964975

SCHEMBL6964975

Cc1nn(-c2ccccc2)c(C)c1N(C#N)C(=O)C(C)c1cccc(C#N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.42
ALDH1A1 P00352 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NOTUM Q6P988 1/20 0.38
GRM5 P41594 1/20 0.37
LMNA P02545 1/20 0.37
GPR139 Q6DWJ6 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
APEX1 P27695 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
RAB9A P51151 2/20 0.35
NR3C1 P04150 1/20 0.35
NPC1 O15118 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964973 0.78 PLK1 (0.40) PLK1ALDH1A1NPSR1TP53TSHR
SCHEMBL6964978 0.78 NPC1 (0.42) ALDH1A1NPSR1TP53TSHRHSD17B10
SCHEMBL6966662 0.72 NPSR1 (0.44) ALDH1A1NPSR1TP53TSHRHSD17B10
SCHEMBL6972133 0.71 MAPT (0.46) PLK1ALDH1A1NPSR1TP53TSHR
SCHEMBL6960209 0.70 PLK1 (0.48) PLK1ALDH1A1NPSR1TP53TSHR
SCHEMBL1990381 0.68 PTGS1 (0.54) ALDH1A1HSD17B10LMNAGPR139KDM4E
SCHEMBL6970481 0.66 MEN1 (0.39) PLK1ALDH1A1NPSR1TP53TSHR
SCHEMBL6965184 0.65 MAPT (0.40) NOTUMNPC1KMT2AMAPT
SCHEMBL27655360 0.64 TDP1 (0.53) ALDH1A1NPSR1TSHRLMNAKDM4E
SCHEMBL11253413 0.64 TDP1 (0.53) ALDH1A1NPSR1TSHRLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed