SCHEMBL6964973

SCHEMBL6964973

CC(=O)N(c1c(C)nn(-c2ccccc2)c1C)C(C#N)c1cccc(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.40
GRM5 P41594 1/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NOTUM Q6P988 1/20 0.38
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
GPR139 Q6DWJ6 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.36
APEX1 P27695 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NR3C1 P04150 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966662 0.76 NPSR1 (0.44) GRM5ALDH1A1LMNATP53TSHR
SCHEMBL6960209 0.72 PLK1 (0.48) PLK1GRM5ALDH1A1LMNATP53
SCHEMBL6972133 0.71 MAPT (0.46) PLK1GRM5ALDH1A1LMNATP53
SCHEMBL6964978 0.70 NPC1 (0.42) GRM5ALDH1A1LMNATP53TSHR
SCHEMBL6970481 0.68 MEN1 (0.39) PLK1GRM5ALDH1A1LMNATP53
SCHEMBL6965184 0.65 MAPT (0.40) NOTUMUBE2MDCUN1D1KMT2AMEN1
SCHEMBL6964956 0.64 L3MBTL1 (0.47) ALDH1A1LMNATSHRNPSR1KMT2A
SCHEMBL4239759 0.64 SLC34A1 (0.51) NPSR1KMT2AMEN1POLBNR3C1
SCHEMBL3834637 0.64 F11 (0.52) PLK1GRM5ALDH1A1TP53TSHR
SCHEMBL6972370 0.63 S1PR1 (0.36) PLK1ALDH1A1LMNATSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed