SCHEMBL6967269

SCHEMBL6967269

Cc1nc(C(C)C)c(Cc2cc(Cl)cc(Cl)c2)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.41
CCR5 P51681 2/20 0.41
HTT P42858 1/20 0.39
PDE5A O76074 1/20 0.36
PDE9A O76083 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
ALDH1A1 P00352 1/20 0.33
TRPV1 Q8NER1 2/20 0.32
ITGA4 P13612 1/20 0.30
TOP2A P11388 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8571054 0.79 CYP1A2 (0.36) ALDH1A1TRPV1TOP2A
SCHEMBL7852268 0.78 CAPN1 (0.47) HTT
SCHEMBL21668150 0.70 ADORA3 (0.33)
SCHEMBL6963010 0.69 TYMS (0.36) HTTALDH1A1TRPV1
SCHEMBL5751774 0.69 CCR2 (0.44) CCR2CCR5HTTPDE5APDE9A
SCHEMBL6973911 0.68 CCR2 (0.41) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL11118144 0.66 LTB4R (0.41) HTTALDH1A1
SCHEMBL8099901 0.62 CCR2 (0.41) CCR2CCR5
SCHEMBL6969892 0.62 CCR2 (0.39) CCR2CCR5
SCHEMBL27967679 0.61 SLC9A1 (0.37) HTTPDE5APDE9APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed