SCHEMBL6973911

SCHEMBL6973911

Cc1nc(C(C)C)c(Cc2cc(Cl)cc(Cl)c2)n1C

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.41
CCR5 P51681 2/20 0.41
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PDE5A O76074 1/20 0.30
PDE9A O76083 1/20 0.30
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099901 0.81 CCR2 (0.41) CCR2CCR5
SCHEMBL6969892 0.81 CCR2 (0.39) CCR2CCR5
SCHEMBL6973294 0.73 CCR2 (0.38) CCR2CCR5
SCHEMBL6965327 0.73 VCP (0.37) CCR2CCR5NPC1RAB9ATDP1
SCHEMBL21668151 0.71
SCHEMBL6966628 0.70 DRD2 (0.34) RECQL
SCHEMBL6960290 0.69 CCR2 (0.43) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL6967269 0.68 CCR2 (0.41) CCR2CCR5PDE5APDE9APDE1A
SCHEMBL10148293 0.67 HTT (0.30)
SCHEMBL5750247 0.66 CCR2 (0.43) CCR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed