SCHEMBL7081541

SCHEMBL7081541

CC(=O)OCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.35
P2RX3 P56373 3/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ALOX12 P18054 1/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PTPN11 Q06124 1/20 0.33
SLC6A9 P48067 1/20 0.33
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973001 0.92 P2RX3 (0.33) IDO1P2RX3CSNK2A2CSNK2BTDP1
SCHEMBL6960281 0.92 PIM1 (0.36) IDO1P2RX3CSNK2A2CSNK2BTDP1
SCHEMBL5852655 0.92 P2RX3 (0.33) P2RX3TDP1KMT2AKDM4EL3MBTL1
SCHEMBL6967425 0.91 ALDH1A1 (0.40) TDP1KMT2ATP53
SCHEMBL6960486 0.91 IDO1 (0.34) IDO1P2RX3CSNK2A2CSNK2BTDP1
SCHEMBL7084851 0.90 P2RX3 (0.35) IDO1P2RX3CSNK2A2CSNK2BTDP1
SCHEMBL6973952 0.90 ENPP2 (0.36) KMT2ATP53SLC6A9MEN1CYP1A2
SCHEMBL6975053 0.90 MEN1 (0.41) P2RX3KMT2ATP53KDM4EMEN1
SCHEMBL7081639 0.88 ALOX12 (0.38) ALOX12KMT2ATP53RXFP1KDM4E
SCHEMBL7081153 0.87 MAPT (0.39) KMT2ATP53RXFP1SLC6A9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed