SCHEMBL6972338

SCHEMBL6972338

CC(=O)OCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.38
GRIN2B Q13224 8/20 0.38
S1PR3 Q99500 4/20 0.35
ENPP2 Q13822 1/20 0.34
LMNA P02545 1/20 0.34
IDO1 P14902 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
PKM P14618 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079752 0.93 GRIN1 (0.37) GRIN1GRIN2BS1PR3ENPP2IDO1
SCHEMBL6960775 0.93 GRIN1 (0.35) GRIN1GRIN2BS1PR3LMNAIDO1
SCHEMBL7086281 0.91 ENPP2 (0.38) GRIN1GRIN2BS1PR3ENPP2LMNA
SCHEMBL6973952 0.91 ENPP2 (0.36) GRIN1GRIN2BENPP2LMNAALDH1A1
SCHEMBL6967425 0.90 ALDH1A1 (0.40) GRIN1GRIN2BS1PR3LMNAALDH1A1
SCHEMBL6969306 0.89 KMT2A (0.39) S1PR3LMNAALDH1A1KMT2APKM
SCHEMBL6972994 0.88 RXFP1 (0.41) LMNAALDH1A1MAPTKMT2A
SCHEMBL7083490 0.88 GRIN1 (0.35) GRIN1GRIN2BS1PR3ENPP2LMNA
SCHEMBL7083459 0.87 GRIN1 (0.35) GRIN1GRIN2BS1PR3LMNAIDO1
SCHEMBL7086202 0.87 LMNA (0.41) GRIN1GRIN2BS1PR3ENPP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed