SCHEMBL6969

SCHEMBL6969

[CH2]Cc1ccccc1NC(=O)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.51
TP53 P04637 2/20 0.48
JAK2 O60674 1/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
KLK7 P49862 1/20 0.48
PARP14 Q460N5 1/20 0.43
ANO1 Q5XXA6 1/20 0.42
PDK1 Q15118 6/20 0.41
PDK2 Q15119 6/20 0.41
PDK3 Q15120 6/20 0.41
PDK4 Q16654 6/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8134750 0.83 AR (0.51) ARTP53JAK2MAPTHTT
SCHEMBL10649798 0.79 AR (0.48) ARTP53JAK2MAPTHTT
SCHEMBL9991690 0.79 TRPV1 (0.54) ARTP53JAK2MAPTHTT
SCHEMBL27401813 0.78 GAA (0.48) MAPTHTTALDH1A1
SCHEMBL1405006 0.78 ALDH1A1 (0.51) ARTP53JAK2MAPTHTT
SCHEMBL12849679 0.78 TRPV1 (0.50) ARTP53JAK2MAPTHTT
SCHEMBL840362 0.77 ALDH1A1 (0.55) HTTNPC1RAB9AHSD17B10ALDH1A1
SCHEMBL5801586 0.77 POLB (0.57) TP53JAK2MAPTHTTKLK7
SCHEMBL7299817 0.74 GAA (0.56) TP53JAK2MAPTHTTKLK7
SCHEMBL1576313 0.74 PDK1 (0.67) TP53JAK2MAPTHTTKLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849911-A Antivirally active heterocyclic azahexane derivatives NOVARTIS FINANCE CORPORATION (US) 1998-12-15 US disclosed
US-5753652-A Antiretroviral hydrazine derivatives NOVARTIS CORPORATION (US) 1998-05-19 US disclosed