SCHEMBL6969301

SCHEMBL6969301

O=C1CCN(C(=O)c2ccc([N+](=O)[O-])c(OCc3ccccc3)c2)c2ccccc2N1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.54
ABCB1 P08183 1/20 0.47
MAPT P10636 7/20 0.46
ALDH1A1 P00352 3/20 0.46
HTT P42858 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
CRBN Q96SW2 2/20 0.45
MAPK1 P28482 2/20 0.45
NPC1 O15118 1/20 0.45
GAA P10253 1/20 0.45
RAB9A P51151 1/20 0.45
THRB P10828 1/20 0.44
VDR P11473 1/20 0.44
PPARG P37231 1/20 0.44
MYC P01106 1/20 0.43
MAX P61244 1/20 0.43
TDP1 Q9NUW8 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955057 0.86 BRD4 (0.57) BRD4MAPTALDH1A1HTTL3MBTL1
SCHEMBL6970210 0.81 BRD4 (0.59) BRD4MAPTALDH1A1HTTL3MBTL1
SCHEMBL6965183 0.77 ABCB1 (0.43) ABCB1MAPTALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL6971322 0.76 ALDH1A1 (0.60) BRD4MAPTALDH1A1HTTL3MBTL1
SCHEMBL6964190 0.76 BRD4 (0.60) BRD4ALDH1A1HTTL3MBTL1SMN1; SMN2
SCHEMBL6966939 0.75 TUBB4A (0.46) BRD4MAPTALDH1A1HTTPOLB
SCHEMBL6954979 0.75 TUBB4A (0.45) BRD4MAPTALDH1A1POLBCRBN
SCHEMBL4909516 0.74 ABCB1 (0.49) ABCB1MAPTSMN1; SMN2MYCMAX
SCHEMBL30082870 0.73 MYC (0.67) ABCB1L3MBTL1POLBMYCMAX
SCHEMBL528177 0.73 MYC (0.67) ABCB1L3MBTL1POLBMYCMAX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed