SCHEMBL6966939

SCHEMBL6966939

COc1cc(C(=O)N2CCC(=O)Nc3cc(C)ccc32)ccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46
TUBA1B P68363 1/20 0.46
TUBA4A P68366 1/20 0.46
TUBB4B P68371 1/20 0.46
TUBB3 Q13509 1/20 0.46
TUBB2A Q13885 1/20 0.46
TUBB8 Q3ZCM7 1/20 0.46
TUBA3E Q6PEY2 1/20 0.46
TUBA1A Q71U36 1/20 0.46
TUBA1C Q9BQE3 1/20 0.46
TUBB6 Q9BUF5 1/20 0.46
TUBB2B Q9BVA1 1/20 0.46
TUBB1 Q9H4B7 1/20 0.46
BRD4 O60885 2/20 0.44
MAPT P10636 6/20 0.43
TDP1 Q9NUW8 3/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954979 0.90 TUBB4A (0.45) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL6955057 0.89 BRD4 (0.57) BRD4MAPTTDP1HPGDNPSR1
SCHEMBL6970424 0.88 ALDH1A1 (0.48) BRD4MAPTTDP1HPGDNPSR1
SCHEMBL6971003 0.83 BRD4 (0.45) BRD4MAPTTDP1HPGDNPSR1
SCHEMBL7355244 0.81 PDE4A (0.47) MAPTNPSR1MEN1CYP3A4CYP2C9
SCHEMBL6970905 0.79 ALDH1A1 (0.47) BRD4MAPTTDP1HPGDNPSR1
SCHEMBL6971322 0.79 ALDH1A1 (0.60) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL6970210 0.77 BRD4 (0.59) BRD4MAPTTDP1HPGDNPSR1
SCHEMBL6970387 0.77 BRD4 (0.52) BRD4MAPTMEN1KMT2AHTT
SCHEMBL6969398 0.76 ALDH1A1 (0.42) MAPTHPGDNPSR1MEN1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed