SCHEMBL6971322

SCHEMBL6971322

COc1cc(C(=O)N2CC(=O)Nc3ccccc32)ccc1[N+](=O)[O-]

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
MAPT P10636 5/20 0.58
TDP1 Q9NUW8 3/20 0.58
HTT P42858 3/20 0.58
MAPK1 P28482 1/20 0.58
NPSR1 Q6W5P4 2/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
HPGD P15428 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
LMNA P02545 1/20 0.56
BRD4 O60885 6/20 0.56
L3MBTL1 Q9Y468 1/20 0.55
TUBB4A P04350 1/20 0.53
TUBB P07437 1/20 0.53
TUBA3C P0DPH7 1/20 0.53
TUBA1B P68363 1/20 0.53
TUBA4A P68366 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955057 0.90 BRD4 (0.57) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL6962591 0.79 HTT (0.71) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL6966939 0.79 TUBB4A (0.46) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL6954979 0.78 TUBB4A (0.45) ALDH1A1MAPTMEN1KMT2AHPGD
SCHEMBL6969301 0.76 BRD4 (0.54) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL6970210 0.76 BRD4 (0.59) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL7348484 0.76 PDE4A (0.53) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL7333735 0.75 AVPR1A (0.66)
SCHEMBL7348149 0.74 PDE4B (0.69) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL9375233 0.73 HTT (1.00) ALDH1A1HTTMAPK1NPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed