SCHEMBL6969333

SCHEMBL6969333

CCn1c(CC#N)nc(C(C)C)c1Sc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HAO1 Q9UJM8 1/20 0.31
DHFR P00374 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
GCGR P47871 1/20 0.31
NOTUM Q6P988 1/20 0.31
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND2 P30279 1/20 0.30
CCND3 P30281 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967795 0.89 ALDH1A1 (0.33) ALDH1A1LMNAMAPT
SCHEMBL6971658 0.88 MAOA (0.36) ALDH1A1HAO1KMT2AMAOAMAOB
SCHEMBL6973627 0.87 MEN1 (0.40) LMNADHFRKMT2AMAOAMAOB
SCHEMBL7080138 0.86 RAB9A (0.34) ALDH1A1LMNAMAPTMAOAMAOB
SCHEMBL7079161 0.86 GRIN1 (0.35) ALDH1A1LMNAKMT2AATM
SCHEMBL6964947 0.86 DHODH (0.34) DHODHALDH1A1LMNAMAPTHAO1
SCHEMBL7086664 0.85 DHODH (0.35) DHODHALDH1A1LMNAMAPTHAO1
SCHEMBL6974771 0.85 DHODH (0.43) DHODHALDH1A1LMNAMAPTHAO1
SCHEMBL6960568 0.84 GRIN1 (0.37) ALDH1A1ATM
SCHEMBL6974210 0.83 DHODH (0.34) DHODHALDH1A1LMNAMAPTHAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed