SCHEMBL6969396

SCHEMBL6969396

CC(C)c1nc(COCc2ccccc2)n(Cc2ccc[nH]c2=O)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.37
P2RX3 P56373 2/20 0.37
KMT2A Q03164 3/20 0.35
RCE1 Q9Y256 1/20 0.33
SLC5A2 P31639 1/20 0.32
CYP2C8 P10632 1/20 0.31
ADAMTS5 Q9UNA0 2/20 0.31
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
VCP P55072 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14439828 0.87 TDP1 (0.40) TDP1KMT2ASLC5A2VCP
SCHEMBL6968197 0.85 P2RX3 (0.36) TDP1P2RX3KMT2ARCE1CYP2C8
SCHEMBL6962617 0.85 P2RX3 (0.35) P2RX3CYP2C8
SCHEMBL6974828 0.84 TDP1 (0.38) TDP1P2RX3KMT2ASLC5A2ADAMTS5
SCHEMBL6967282 0.83 TDP1 (0.32) TDP1KMT2AVCP
SCHEMBL27412267 0.83 TDP1 (0.36) TDP1P2RX3KMT2ARCE1SLC5A2
SCHEMBL6972460 0.82 P2RX3 (0.36) TDP1P2RX3VCP
SCHEMBL5853114 0.82 TDP1 (0.37) TDP1SLC5A2VCP
SCHEMBL6966496 0.82 VCP (0.37) TDP1SLC5A2ADAMTS5MMP2MMP13
SCHEMBL6965896 0.81 VCP (0.36) TDP1SLC5A2ADAMTS5MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed