SCHEMBL6972460

SCHEMBL6972460

COc1ncccc1Cn1c(COCc2ccccc2)nc(C(C)C)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.36
TDP1 Q9NUW8 1/20 0.34
PDE1A P54750 5/20 0.33
PDE1B Q01064 5/20 0.33
PDE1C Q14123 5/20 0.33
KDM1A O60341 3/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
DHODH Q02127 1/20 0.32
VCP P55072 1/20 0.32
TP53 P04637 2/20 0.31
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
AVPR1A P37288 1/20 0.30
ENPP2 Q13822 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967282 0.91 TDP1 (0.32) TDP1DHODHVCPTP53MAPT
SCHEMBL14439828 0.87 TDP1 (0.40) TDP1DHODHVCPTP53MAPT
SCHEMBL5853114 0.87 TDP1 (0.37) TDP1DHODHVCPTP53MAPT
SCHEMBL6960433 0.86 TDP1 (0.34) P2RX3TDP1VCPTP53MAPT
SCHEMBL6957630 0.85 DHODH (0.39) TDP1DHODHTP53MAPT
SCHEMBL14439857 0.85 DHODH (0.39) TDP1DHODHTP53MAPT
SCHEMBL6960939 0.83 TP53 (0.35) P2RX3TDP1VCPTP53MAPT
SCHEMBL6966496 0.83 VCP (0.37) TDP1DHODHVCPTP53MAPT
SCHEMBL6969396 0.82 TDP1 (0.37) P2RX3TDP1VCP
SCHEMBL14439830 0.82 TP53 (0.39) TDP1DHODHVCPTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed