SCHEMBL6974828

SCHEMBL6974828

CC(C)c1nc(COCc2ccccc2)n(Cc2ccc(=O)[nH]c2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
P2RX3 P56373 2/20 0.35
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.33
SLC5A2 P31639 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
ADAMTS5 Q9UNA0 2/20 0.32
VCP P55072 1/20 0.32
MMP2 P08253 1/20 0.32
MMP13 P45452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14439828 0.89 TDP1 (0.40) TDP1KMT2AMAPTSMN1; SMN2L3MBTL1
SCHEMBL6957630 0.85 DHODH (0.39) TDP1ALDH1A1HTTMAPTPOLB
SCHEMBL14439857 0.85 DHODH (0.39) TDP1ALDH1A1HTTMAPTPOLB
SCHEMBL5853114 0.85 TDP1 (0.37) TDP1ALDH1A1MAPTKDM4ETP53
SCHEMBL6969568 0.85 P2RX3 (0.37) TDP1ALDH1A1HTTMEN1KMT2A
SCHEMBL6962868 0.85 P2RX3 (0.35) TDP1ALDH1A1HTTP2RX3GAA
SCHEMBL6969396 0.84 TDP1 (0.37) TDP1KMT2AP2RX3SLC5A2ADAMTS5
SCHEMBL7087497 0.83 P2RX3 (0.36) TDP1ALDH1A1HTTMEN1KMT2A
SCHEMBL6966496 0.83 VCP (0.37) TDP1MAPTSMN1; SMN2L3MBTL1TP53
SCHEMBL27397423 0.82 TDP1 (0.37) TDP1ALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed