SCHEMBL6972014

SCHEMBL6972014

O=C(CC(=O)C(F)(F)F)c1nc2cccc(F)c2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 3/20 0.41
PLOD3 O60568 2/20 0.40
PLOD1 Q02809 2/20 0.40
AKR1A1 P14550 1/20 0.39
AKR1B1 P15121 1/20 0.39
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOB P27338 2/20 0.35
NAAA Q02083 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
RECQL P46063 1/20 0.34
RIPK1 Q13546 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CD38 P28907 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979211 0.79 RAB9A (0.58) RAB9ANPC1HPGDSMN1; SMN2MAOB
SCHEMBL6979685 0.78 GAA (0.47) PLOD2PLOD3PLOD1AKR1A1AKR1B1
SCHEMBL7960065 0.76 AKR1A1 (0.43) AKR1A1AKR1B1RAB9ANPC1HPGD
SCHEMBL19691127 0.75 DYRK1A (0.43) AKR1A1AKR1B1RAB9ANPC1SMN1; SMN2
SCHEMBL6977213 0.75 GAA (0.40) AKR1A1AKR1B1RAB9ANPC1SMN1; SMN2
SCHEMBL6981786 0.73 DYRK1A (0.49) PLOD2PLOD3PLOD1AKR1A1AKR1B1
SCHEMBL6982879 0.73 PDPK1 (0.49) PLOD2RAB9ANPC1HPGDSMN1; SMN2
SCHEMBL6969298 0.71 STING1 (0.39) PLOD2PLOD3PLOD1MAOBHSD17B1
SCHEMBL8643935 0.71 PLOD2 (0.55) PLOD2PLOD3PLOD1RAB9ANPC1
Trifluoroacetic Acid SCHEMBL29974297 0.70 SMN1; SMN2 (0.41) AKR1A1AKR1B1RAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed