SCHEMBL6969298

SCHEMBL6969298

Cc1cc2nc(C(=O)CC(=O)C(F)(F)F)sc2cc1F

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 2/20 0.39
PLOD2 O00469 2/20 0.36
MAOB P27338 10/20 0.36
PLOD3 O60568 1/20 0.35
PLOD1 Q02809 1/20 0.35
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
GAA P10253 1/20 0.33
PPOX P50336 2/20 0.33
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975865 0.81 TP53 (0.51) MAOBGAA
SCHEMBL6982879 0.79 PDPK1 (0.49) PLOD2MAOBGAA
SCHEMBL6981786 0.79 DYRK1A (0.49) PLOD2MAOBPLOD3PLOD1
SCHEMBL6979450 0.78 GAA (0.41) STING1MAOBHSD17B1HSD17B2GAA
SCHEMBL6983733 0.75 DYRK1A (0.48) MAOBGAA
SCHEMBL6979367 0.75 MAPT (0.57) MAOBHSD17B1HSD17B2
SCHEMBL6979211 0.74 RAB9A (0.58) MAOBHSD17B1HSD17B2GAA
SCHEMBL6979685 0.71 GAA (0.47) PLOD2PLOD3PLOD1GAA
SCHEMBL6972014 0.71 PLOD2 (0.41) PLOD2MAOBPLOD3PLOD1HSD17B1
SCHEMBL6975976 0.71 ACP1 (0.47) MAOBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed