SCHEMBL6972194

SCHEMBL6972194

CC(=O)Nc1ccc(Cn2c(CO)nc(C(C)C)c2Sc2cc(Cl)cc(Cl)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RAB9A P51151 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 3/20 0.41
TP53 P04637 2/20 0.41
P2RX3 P56373 5/20 0.38
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
USP1 O94782 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NOD1 Q9Y239 1/20 0.36
NLRP3 Q96P20 1/20 0.36
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959976 0.90 P2RX3 (0.39) NPC1LMNASMN1; SMN2RAB9AGAA
SCHEMBL14439855 0.86 TDP1 (0.33) P2RX3
SCHEMBL14439870 0.85 P2RX3 (0.43) LMNARAB9AGAAMAPTTP53
Acetamide SCHEMBL6972197 0.85 TDP1 (0.41) LMNASMN1; SMN2MAPTP2RX3MEN1
SCHEMBL6971451 0.85 HSP90B1 (0.33) SMN1; SMN2TP53P2RX3KDM4EALDH1A1
SCHEMBL6966848 0.84 TDP1 (0.42) GAAMAPTTP53MEN1KMT2A
SCHEMBL14439868 0.84 DCTPP1 (0.34) P2RX3
SCHEMBL5852651 0.83 KCNH2 (0.35) MEN1HTTKMT2A
Carbamic Acid SCHEMBL667612 0.82 PIM1 (0.36) P2RX3MEN1KMT2A
SCHEMBL6961345 0.82 L3MBTL1 (0.39) NPC1SMN1; SMN2RAB9AP2RX3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed