SCHEMBL6961345

SCHEMBL6961345

CC(C)c1nc(CO)n(Cc2ccc([N+](=O)[O-])cc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
AR P10275 2/20 0.37
DHFR P00374 1/20 0.35
TYMS P04818 1/20 0.35
TBXA2R P21731 1/20 0.35
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
NR2F2 P24468 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SRC P12931 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
NOX4 Q9NPH5 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969108 0.92 TSHR (0.38) L3MBTL1MEN1KMT2AARDHFR
SCHEMBL6970372 0.91 CCR2 (0.43) L3MBTL1MEN1KMT2AKDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL6969480 0.90 CCR2 (0.43) L3MBTL1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL14439866 0.87 L3MBTL1 (0.38) L3MBTL1MEN1KMT2AARDHFR
SCHEMBL14439855 0.86 TDP1 (0.33) P2RX3
SCHEMBL6962314 0.85 L3MBTL1 (0.36) L3MBTL1MEN1KMT2AARDHFR
SCHEMBL6971451 0.85 HSP90B1 (0.33) KDM4ESMN1; SMN2P2RX3ALDH1A1
SCHEMBL6966848 0.84 TDP1 (0.42) MEN1KMT2AKDM4EALDH1A1POLB
SCHEMBL14439868 0.84 DCTPP1 (0.34) P2RX3
SCHEMBL6964071 0.84 ALDH1A1 (0.35) MEN1KMT2AKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed