SCHEMBL6973430

SCHEMBL6973430

COc1ccc(COCC(c2cccnc2)c2nc(C(C)C)c(Sc3cc(Cl)cc(Cl)c3)[nH]2)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
ALOX15 P16050 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
TACR1 P25103 2/20 0.31
TBXAS1 P24557 2/20 0.31
KCNA5 P22460 2/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
RORC P51449 2/20 0.30
THRB P10828 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962307 0.78 CYP1A2 (0.35) ALDH1A1KCNA5LMNACYP2C9
SCHEMBL6973659 0.73 MEN1 (0.34) ALDH1A1HSD17B10TBXAS1LMNAMAPT
SCHEMBL6973428 0.72 GABRA1 (0.36) USP2ALDH1A1GAAALOX15RECQL
SCHEMBL5852619 0.72 TACR1 (0.34) TACR1
SCHEMBL6973717 0.72 LMNA (0.35) ALDH1A1LMNAMAPTCYP2C9
SCHEMBL6971891 0.71 ALDH1A1 (0.37) ALDH1A1TACR1
SCHEMBL6971468 0.70 HRH4 (0.36) ALDH1A1TACR1
SCHEMBL6973278 0.70 MEN1 (0.35) ALDH1A1HSD17B10TBXAS1LMNARORC
SCHEMBL7085227 0.69 IDO1 (0.31) MAPT
SCHEMBL8349719 0.68 KCNA5 (0.37) ALDH1A1KCNA5CYP19A1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed