SCHEMBL6962307

SCHEMBL6962307

COc1ccc(COCc2nc(C(C)C)c(Sc3cc(Cl)cc(Cl)c3)[nH]2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP2E1 P05181 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C8 P10632 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2B6 P20813 2/20 0.35
CYP2C19 P33261 2/20 0.35
DHFR P00374 2/20 0.35
DHODH Q02127 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CCNB2 O95067 1/20 0.32
CCNE2 O96020 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCND1 P24385 1/20 0.32
CCNE1 P24864 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973717 0.91 LMNA (0.35) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL14001863 0.81 HSP90B1 (0.31)
SCHEMBL6964698 0.81 LMNA (0.36) CYP1A2CYP3A4CYP2C9CYP2C19HCAR2
SCHEMBL6971891 0.80 ALDH1A1 (0.37) DHODHHCAR2MMP13ALDH1A1TDP1
SCHEMBL5029294 0.79 DHFR (0.41) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL6973531 0.79 CNR2 (0.39) LMNARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL6971468 0.78 HRH4 (0.36) ALDH1A1TDP1REN
SCHEMBL6973430 0.78 USP2 (0.33) CYP2C9LMNAALDH1A1KCNA5
SCHEMBL6559757 0.78 TDP1 (0.36) DHFRKDM4ETDP1
SCHEMBL6964520 0.77 DHODH (0.34) CYP3A4DHFRDHODHCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed