SCHEMBL14439826

SCHEMBL14439826

CC(C)c1nc(COCc2ccccc2)[nH]c1Sc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
DHFR P00374 3/20 0.38
CAPN1 P07384 1/20 0.36
VCP P55072 1/20 0.36
ALDH1A1 P00352 2/20 0.33
PDE9A O76083 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
SLC6A4 P31645 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
ALOX5 P09917 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5029294 0.89 DHFR (0.41) DHFRALDH1A1HCAR2
SCHEMBL6964698 0.89 LMNA (0.36) PDE9APDE1APDE1BPDE1CSLC6A4
SCHEMBL6974600 0.88 TSHR (0.33) TSHRCAPN1VCPALDH1A1PDE9A
SCHEMBL5852619 0.88 TACR1 (0.34) TSHRCAPN1VCPPDE9APDE1A
SCHEMBL14439851 0.87 TSHR (0.41) TSHRCAPN1VCPALDH1A1PDE9A
SCHEMBL14002290 0.84 DHFR (0.36) DHFRALDH1A1ALOX5
SCHEMBL6973717 0.79 LMNA (0.35) DHFRALDH1A1TOP2AHCAR2
SCHEMBL6971891 0.79 ALDH1A1 (0.37) CAPN1ALDH1A1HCAR2
SCHEMBL4893143 0.79 TSHR (0.43) TSHRCAPN1VCPALDH1A1PDE9A
SCHEMBL6962307 0.77 CYP1A2 (0.35) DHFRALDH1A1CA1CA2HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed