SCHEMBL6973746

SCHEMBL6973746

CNC(=O)OCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
ENPP2 Q13822 1/20 0.36
CACNA1I Q9P0X4 1/20 0.35
S1PR3 Q99500 4/20 0.35
CYP3A4 P08684 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078901 0.94 ALDH1A1 (0.40) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL6973275 0.91 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ACACNA1IS1PR3
SCHEMBL6961504 0.91 ENPP2 (0.35) ALDH1A1MEN1KMT2ALMNAHTT
SCHEMBL6973878 0.90 MEN1 (0.35) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL6967367 0.90 ENPP2 (0.39) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7080182 0.90 MAPT (0.35) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL6957033 0.90 ADRA1D (0.37) ALDH1A1MEN1KMT2ACACNA1IS1PR3
SCHEMBL6964229 0.90 TOP2A (0.41) ENPP2S1PR3CYP3A4
SCHEMBL7086281 0.87 ENPP2 (0.38) MAPTLMNAENPP2S1PR3CYP3A4
SCHEMBL6969211 0.85 KMT2A (0.34) ALDH1A1MEN1KMT2ACACNA1IS1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed