SCHEMBL7086281

SCHEMBL7086281

CNC(=O)OCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.38
GRIN1 Q05586 6/20 0.37
GRIN2B Q13224 6/20 0.37
S1PR3 Q99500 4/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967367 0.94 ENPP2 (0.39) ENPP2GRIN1GRIN2BS1PR3HDAC1
SCHEMBL6972338 0.91 GRIN1 (0.38) ENPP2GRIN1GRIN2BS1PR3LMNA
SCHEMBL6967603 0.91 ENPP2 (0.40) ENPP2GRIN1GRIN2BLMNACYP3A4
SCHEMBL7083490 0.90 GRIN1 (0.35) ENPP2GRIN1GRIN2BS1PR3LMNA
SCHEMBL7078901 0.90 ALDH1A1 (0.40) ENPP2GRIN1GRIN2BS1PR3HDAC1
SCHEMBL6964229 0.90 TOP2A (0.41) ENPP2S1PR3CYP3A4
SCHEMBL6974914 0.88 RXFP1 (0.39) LMNAMAPT
SCHEMBL6973746 0.87 ALDH1A1 (0.37) ENPP2S1PR3HDAC1HDAC3HDAC4
SCHEMBL6960775 0.86 GRIN1 (0.35) GRIN1GRIN2BS1PR3LMNAMAPT
SCHEMBL7086602 0.85 TOP2A (0.34) ENPP2LMNACYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed