SCHEMBL7080182

SCHEMBL7080182

CNC(=S)OCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
S1PR3 Q99500 4/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
PKM P14618 2/20 0.32
KMT2A Q03164 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
SRC P12931 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRA5 P31644 1/20 0.31
TP53 P04637 1/20 0.31
MEN1 O00255 1/20 0.31
HIF1A Q16665 1/20 0.31
P2RX3 P56373 1/20 0.31
SLC16A3 O15427 1/20 0.31
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085898 0.94 ALDH1A1 (0.37) S1PR3HTTSMN1; SMN2PKMKMT2A
SCHEMBL6961663 0.91 P2RX3 (0.31) P2RX3
SCHEMBL6974277 0.90 GRIN1 (0.34) S1PR3HTTSMN1; SMN2PKMSRC
SCHEMBL6973746 0.90 ALDH1A1 (0.37) MAPTS1PR3HTTCACNA1IKMT2A
SCHEMBL6976430 0.90 HTT (0.34) S1PR3HTTSMN1; SMN2SRCALDH1A1
SCHEMBL6973275 0.87 ALDH1A1 (0.36) S1PR3CACNA1IKMT2AALDH1A1GABRA1
SCHEMBL7083490 0.87 GRIN1 (0.35) S1PR3HTTSMN1; SMN2KMT2ASRC
SCHEMBL6957033 0.86 ADRA1D (0.37) S1PR3CACNA1IKMT2AALDH1A1GABRA1
SCHEMBL6961267 0.85 ALDH1A1 (0.34) MAPTHTTSMN1; SMN2ALDH1A1TP53
SCHEMBL6962639 0.84 RXFP1 (0.37) MAPTMAPK1HTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed