SCHEMBL6964229

SCHEMBL6964229

CNC(=O)OCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.41
TOP2B Q02880 2/20 0.41
CYP3A4 P08684 3/20 0.40
NAMPT P43490 1/20 0.36
S1PR3 Q99500 1/20 0.36
ENPP2 Q13822 1/20 0.36
EPHX1 P07099 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086281 0.90 ENPP2 (0.38) CYP3A4S1PR3ENPP2
SCHEMBL7078901 0.90 ALDH1A1 (0.40) CYP3A4S1PR3ENPP2
SCHEMBL6969306 0.90 KMT2A (0.39) CYP3A4S1PR3L3MBTL1
SCHEMBL6974505 0.90 TOP2A (0.42) TOP2ATOP2BENPP2EPHX1
SCHEMBL6967367 0.90 ENPP2 (0.39) TOP2ATOP2BCYP3A4S1PR3ENPP2
SCHEMBL6973746 0.90 ALDH1A1 (0.37) CYP3A4S1PR3ENPP2
SCHEMBL6976430 0.89 HTT (0.34) CYP3A4S1PR3
SCHEMBL7086385 0.89 TLR7 (0.35) CYP3A4S1PR3L3MBTL1
SCHEMBL6974914 0.88 RXFP1 (0.39)
SCHEMBL6973129 0.84 ALDH1A1 (0.35) CYP3A4S1PR3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed