SCHEMBL6975780

SCHEMBL6975780

Cc1ccc(-c2c(C(N)=O)ccnc2N2CCOCC2)cc1NC(=O)c1cccc(OC2CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 3/20 0.43
RAF1 P04049 6/20 0.41
BRAF P15056 6/20 0.41
PIK3CA P42336 1/20 0.41
MTOR P42345 1/20 0.41
PIK3CG P48736 1/20 0.41
ATR Q13535 1/20 0.41
AURKB Q96GD4 1/20 0.41
CHEK2 O96017 1/20 0.40
MAPK14 Q16539 4/20 0.40
OPRK1 P41145 1/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NEK2 P51955 1/20 0.39
RAB9A P51151 1/20 0.39
SMO Q99835 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973788 0.96 TBK1 (0.44) TBK1RAF1BRAFPIK3CAMTOR
SCHEMBL6979964 0.93 CHEK2 (0.46) TBK1RAF1BRAFPIK3CAMTOR
SCHEMBL6972614 0.89 TBK1 (0.47) TBK1RAF1BRAFPIK3CAMTOR
SCHEMBL6975779 0.82 MAPK14 (0.58) RAF1BRAFMAPK14SMO
SCHEMBL6969091 0.80 MAPK14 (0.42) MAPK14ALDH1A1SMN1; SMN2SMOTSHR
SCHEMBL6476766 0.79 OPRK1 (0.59) RAF1BRAFMAPK14OPRK1ALDH1A1
SCHEMBL2972096 0.79 OPRK1 (0.58) RAF1BRAFMAPK14OPRK1SMO
SCHEMBL7804552 0.78 OPRK1 (0.54) MAPK14OPRK1ALDH1A1SMN1; SMN2RAB9A
SCHEMBL6973786 0.78 MAPK14 (0.57) RAF1BRAFMAPK14SMO
SCHEMBL6477083 0.76 MAPK14 (0.54) BRAFMAPK14OPRK1SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115707-B1 BENZAMIDE DERIVATIVES AND THER USE AS CYTOKINE INHIBITORS ASTRAZENECA AB (SE) 2003-11-12 EP disclosed