SCHEMBL6973788

SCHEMBL6973788

Cc1ccc(-c2c(C(N)=O)ccnc2N2CCOCC2)cc1NC(=O)c1cccc(OC2CCN(C(=O)OC(C)(C)C)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 3/20 0.44
PIK3CD O00329 1/20 0.41
RAF1 P04049 4/20 0.40
BRAF P15056 4/20 0.40
CHEK2 O96017 1/20 0.39
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
PIK3CG P48736 1/20 0.39
ATR Q13535 1/20 0.39
AURKB Q96GD4 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK14 Q16539 4/20 0.38
SMO Q99835 1/20 0.38
OPRK1 P41145 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975780 0.96 TBK1 (0.43) TBK1RAF1BRAFCHEK2PIK3CA
SCHEMBL6979964 0.89 CHEK2 (0.46) TBK1RAF1BRAFCHEK2PIK3CA
SCHEMBL6972614 0.85 TBK1 (0.47) TBK1RAF1BRAFPIK3CAMTOR
SCHEMBL6973786 0.82 MAPK14 (0.57) RAF1BRAFMAPK14SMO
SCHEMBL6533594 0.80 OPRK1 (0.56) RAF1BRAFALDH1A1MAPK14SMO
SCHEMBL2979241 0.79 OPRK1 (0.55) RAF1BRAFALDH1A1MAPK14SMO
SCHEMBL6969091 0.79 MAPK14 (0.42) ALDH1A1SMN1; SMN2MAPK14SMOTSHR
SCHEMBL7806472 0.79 OPRK1 (0.51) TBK1ALDH1A1SMN1; SMN2MAPK14SMO
SCHEMBL6975779 0.78 MAPK14 (0.58) RAF1BRAFMAPK14SMO
SCHEMBL6973782 0.76 TBK1 (0.36) TBK1RAF1BRAFCHEK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115707-B1 BENZAMIDE DERIVATIVES AND THER USE AS CYTOKINE INHIBITORS ASTRAZENECA AB (SE) 2003-11-12 EP disclosed