SCHEMBL6977890

SCHEMBL6977890

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4cccc5ccccc45)c32)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 4/20 0.46
PREP P48147 1/20 0.40
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
GAA P10253 2/20 0.37
POLB P06746 1/20 0.37
USP30 Q70CQ3 1/20 0.36
RAB9A P51151 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
HTR7 P34969 1/20 0.36
PGGT1B P53609 1/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982500 0.90 SLC16A3 (0.48) SLC16A3PREPCHRM2CHRM4CHRM1
SCHEMBL6977188 0.88 NR3C1 (0.48) GAAUSP30
SCHEMBL6985322 0.87 GAA (0.41) GAARAB9ATSHRMEN1ALDH1A1
SCHEMBL6985835 0.87 SLC16A3 (0.42) SLC16A3PREPFNTAFNTBGAA
SCHEMBL6982163 0.86 SLC16A3 (0.45) SLC16A3GAATSHRMEN1USP2
SCHEMBL6977885 0.85 NR3C1 (0.48) TSHR
SCHEMBL6978217 0.84 SLC16A3 (0.42) SLC16A3TSHRMEN1ALDH1A1HPGD
SCHEMBL6986981 0.84 MCL1 (0.40) GAADPP8DPP9MEN1ALDH1A1
SCHEMBL6985566 0.84 PARP14 (0.40) RAB9ADPP8DPP9TSHRMEN1
SCHEMBL6985749 0.83 ALDH1A1 (0.48) GAAMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed