SCHEMBL6982500

SCHEMBL6982500

NCc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4cccc5ccccc45)c32)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 5/20 0.48
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
GAA P10253 2/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.38
HTR7 P34969 3/20 0.38
MCL1 Q07820 1/20 0.37
KCNA5 P22460 1/20 0.37
F10 P00742 1/20 0.37
PREP P48147 1/20 0.36
HTR1A P08908 1/20 0.36
HTR2B P41595 1/20 0.36
HTR6 P50406 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977890 0.90 SLC16A3 (0.46) SLC16A3CHRM2CHRM4CHRM1CHRM3
SCHEMBL6984843 0.86 GAA (0.43) GAAPOLBTSHRHTR6
SCHEMBL6982493 0.83 NR3C1 (0.50) TSHRHTR6
SCHEMBL6981764 0.82 METAP2 (0.42) SLC16A3GAA
SCHEMBL6982743 0.79 F2 (0.42) GAAF10
SCHEMBL6981837 0.79 AVPR2 (0.39) GAA
SCHEMBL6977188 0.78 NR3C1 (0.48) GAAMCL1
SCHEMBL6984787 0.77 ATM (0.48) POLB
SCHEMBL6985835 0.76 SLC16A3 (0.42) SLC16A3GAATSHRPREP
SCHEMBL6985322 0.76 GAA (0.41) GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed